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Experiments

Compound Investigated event Experiment type Concentration Cell line Organism Animal model Stat protein Details
Brevilin A Influence on protein upon cytokine treatment Western Blot 10.00 µM HEK293T Homo sapiens pTyr705-STAT3
Brevilin A Influence on protein upon cytokine treatment Western Blot 10.00 µM HEK293T Homo sapiens STAT3
Brevilin A Influence on protein upon cytokine treatment Western Blot 10.00 µM HEK293T Homo sapiens
Brevilin A Influence on protein upon cytokine treatment RT-PCR 10.00 µM HEK293T Homo sapiens
Brevilin A Influence on protein upon cytokine treatment RT-PCR 10.00 µM HEK293T Homo sapiens
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 10.00 µM HEK293T Homo sapiens pTyr705-STAT3
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 15.00 µM HEK293T Homo sapiens pTyr705-STAT3
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 10.00 µM HEK293T Homo sapiens STAT3
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 15.00 µM HEK293T Homo sapiens STAT3
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 10.00 µM HEK293T Homo sapiens
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 15.00 µM HEK293T Homo sapiens
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 10.00 µM HEK293T Homo sapiens
Brevilin A Influence on JAK2-JH1 overexpressed protein Western Blot 15.00 µM HEK293T Homo sapiens
Brevilin A Influence on c-Src overexpressed protein Western Blot 15.00 µM HEK293T Homo sapiens
Brevilin A Influence on c-Src overexpressed protein Western Blot 15.00 µM HEK293T Homo sapiens
Brevilin A Influence on c-Src overexpressed protein Western Blot 15.00 µM HEK293T Homo sapiens
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 10.00 µM HEK293T Homo sapiens pTyr705-STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 20.00 µM HEK293T Homo sapiens pTyr705-STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 40.00 µM HEK293T Homo sapiens pTyr705-STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 80.00 µM HEK293T Homo sapiens pTyr705-STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 10.00 µM HEK293T Homo sapiens STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 20.00 µM HEK293T Homo sapiens STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 40.00 µM HEK293T Homo sapiens STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 80.00 µM HEK293T Homo sapiens STAT3
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 10.00 µM HEK293T Homo sapiens
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 20.00 µM HEK293T Homo sapiens
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 40.00 µM HEK293T Homo sapiens
Brevilin A Influence on kinase activity (kinase assay) Tyk2-JH1 kinase domain Western Blot 80.00 µM HEK293T Homo sapiens
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens pTyr701-STAT1
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens STAT1
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 5.00 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 7.50 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 10.00 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 12.50 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 17.50 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 20.00 µM HEK293T (JAK1-JH1) Homo sapiens pTyr705-STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 5.00 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 7.50 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 10.00 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 12.50 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 15.00 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 17.50 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Measurement of IC50 value JAKs-JH1 truncated kinases Western Blot 20.00 µM HEK293T (JAK1-JH1) Homo sapiens STAT3
Brevilin A Influence on protein overexpression Western Blot 15.00 µM HEK293T (JAK2-JH1) Homo sapiens pTyr705-STAT3